Search Result "first-pass effect"


Visualization of First-Pass Drug Metabolism of Terfenadine by MALDIImaging Mass Spectrometry

Journal: Drug Metabolism Letters
Volume: 2 Issue: 1 Year: 2008 Page: 1-4
Author(s): Yunsheng Hsieh, Jiwen Chen, Ian Knemeyer, Lee Crossman, Walter A. Korfmacher

Identification of a Novel Intestinal First Pass Metabolic Pathway: NQO1 Mediated Quinone Reduction and Subsequent Glucuronidation

Journal: Current Drug Metabolism
Volume: 8 Issue: 2 Year: 2007 Page: 137-149
Author(s): Haiping Hao, Guangji Wang, Nan Cui, Jing Li, Lin Xie, Zuoqi Ding

The Use of 1-Aminobenzotriazole in Differentiating the Role of CYPMediated First Pass Metabolism and Absorption in Limiting Drug Oral Bioavailability: A Case Study

Journal: Drug Metabolism Letters
Volume: 2 Issue: 2 Year: 2008 Page: 120-124
Author(s): Ayman F. El-Kattan, Julie Poe, Lisa Buchholz, Hayden V. Thomas, Joanne Brodfuehrer, Alan Clark

Maximal Inhibition of Intestinal First-Pass Metabolism as a Pragmatic Indicator of Intestinal Contribution to the Drug-Drug Interactions for CYP3A4 Cleared Drugs

Journal: Current Drug Metabolism
Volume: 8 Issue: 7 Year: 2007 Page: 685-693
Author(s): Aleksandra Galetin, Laura K. Hinton, Howard Burt, R. Scott Obach, J. Brian Houston

Mathematical Model of Low-Pass Filters

Journal: Recent Patents on Engineering
Volume: 5 Issue: 2 Year: 2011 Page: 155-162
Author(s): Jose de Jesus Rubio, Diana M. Vazquez, Jaime Pacheco, Vicente Garcia

Intestinal Transport as a Potential Determinant of Drug Bioavailability

Journal: Current Clinical Pharmacology
Volume: 8 Issue: 3 Year: 2013 Page: 247-255
Author(s): Andromeda M. Nauli, Surya M. Nauli

Research Article

Molecular Dynamics (MD) Simulation of Multi-pass Nanometric Machining – The Effect of Machining Conditions

Journal: Current Nanoscience
Volume: 13 Issue: 1 Year: 2017 Page: 21-30
Author(s): Akinjide Olufemi Oluwajobi,Xun Chen

Research Article

Design, Synthesis, and Pharmacokinetic Evaluation of O-Carbamoyl Tizoxanide Prodrugs

Journal: Medicinal Chemistry
Volume: 16 Issue: 0 Year: 2020 Page: 1-12
Author(s): Xi He,Wenjun Hu,Fanhua Meng,Xingzhou Li

Review Article

Transcending the Cutaneous Barrier Through Nanocarrier Exploration for Passive Delivery of Anti-hypertensive Drugs: A Critical Review

Journal: Recent Patents on Nanotechnology
Volume: 14 Issue: 3 Year: 2020 Page: 193-209
Author(s): Lalit Kumar,Puneet Utreja

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